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Jianhui Huang——Professor

Office 504C, Building 24, Tianjin University
School of Pharmaceutical Science and Technology
Group weblink
Education Experience
2003-2006 Doctor of Philosophy  Chemistry University of York, UK
1996-2000 Bachelor of Science Chemistry Hu'nan University
Professional Experience
2000-2003 Research Associate Tianjin Institute of Pharmaceutical Research,China
2007-2010 Post-doctorial Research Associate University of Sheffield and GlaxoSmithKlein
2010-2017 Associate Professor Tianjin University, China
2017- Professor Tianjin University
Research Area

The research of the Huang group encompasses three main areas:  1) Studies towards the synthesis of heterocycles via transition metal catalysis, 


2) Design and synthesis of useful active pharmaceutical ingredients, and 

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3) Late-stage functionalization of drug molecules and other materials.

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Honors and Awards
Thieme Chemistry Journal Award, 2017
Best Publication Award, HSP, Tianjin University, 2015
钌催化下的2-(3-溴苯基)吡啶类衍生物的合成, 2015031900635430, 黄剑辉、于庆贞、胡乐安、王悦、赵康, 2016.09
2-取代乙烯醇甲酸酯类衍生物的制备方法, 201210441980X, 黄剑辉、杨丹、丁诗璇、赵康, 2014.07
3-羟基-2-烷氧基-3-苯基异吲哚-1(2H)-酮类衍生物的制备方法, 2013102117068, 黄剑辉、刘伟东、朱怡、于庆贞、张娜娜, 2015.07
Highlighted Publications
R. Zhu; Z. Liu; J. Chen; X. Xiong; Y. Wang; L. Huang; J. Bai; Y. Dang; J. Huang ” The preparation of thioanisole biscarbanion and C–H lithiation/annulation reactions for the access of five-membered heterocycles” Org. Lett., 2018, 3161-3165.
Y. Wang; J. Liu; L. Huang; R. Zhu; X. Huang; R. Moir and J. Huang "KOtBu-catalyzed lithiation of PMDTA and the direct functionalization of bridged alkenens under mild conditions." Chem. Commun., 2017, 53, 4589-4592.
Z. Chen; L. Hu; F. Zeng; R. Zhu; S. Zheng; Q. Yu and J. Huang "Selective mono-alkylation of N-methoxybenzamides." Chem. Commun., 2017, 53, 4258-4261.
Q. Yu; L. Hu; Y. Wang; S. Zheng; J. Huang "Directed meta-selective bromination of arenes with ruthenium catalysts." Angew. Chem. Int. Ed., 2015, 54, 15284-15288.
W. Liu; Q. Yu; L. Hu; J. Huang "Modular synthesis of dihydro-isoquinolines: palladium-catalyzed sequential C(sp2)-H and C(sp3)-H bond activation." Chem. Sci., 2015, 6, 5768-5772.
Zhong, H.; Yang, D.; Wang, S.; Huang, J. Pd-catalyzed synthesis of isoquinolinones and analogues via C-H and N-H bonds double activation. Chem. Commun. 2012, 48, 3236.
ResearcherID Publications
Year Title Author(s) Source Volume
2009 Lithiation-electrophilic trapping of N-sulfonyl-activated ethylene aziridines Huang, Jianhui; Moore, Stephen P.; O’Brien, Peter; et al. Organic & Biomolecular Chemistry 7
2009 A divergent strategy to the withasomnines Foster, Robert S.; Huang, Jianhui; Vivat, Jerome F.; et al. Organic & Biomolecular Chemistry 7
2009 A direct route to triazole boronic esters and their application in the synthesis of small molecule arrays Huang, Jianhui; Macdonald, Simon J. F.; Cooper, Anthony W. J.; et al. Tetrahedron Letters 50
2009 A cycloaddition route to novel triazole boronic esters Huang, Jianhui; Macdonald, Simon J. F.; Harrity, Joseph P. A. Chemical Communications
2010 Syntheses of N-Alkylated Carbazolones via Pd(OAc)(2)-Mediated Intramolecular Coupling of N-Substituted 3-(Arylamino)cyclohex-2-enones Bi, Wenying; Yun, Xiliu; Fan, Yanfeng; et al. Synlett
2010 A borylative cyclisation towards indole boronic esters Huang, Jianhui; Macdonald, Simon J. F.; Harrity, Joseph P. A. Chemical Communications 46
2011 Synthesis of Coumestan Derivatives via FeCl3-Mediated Oxidative Ring Closure of 4-Hydroxy Coumarins Tang, Lina; Pang, Yongle; Yan, Qiao; et al. Journal of Organic Chemistry 76
2011 Synthesis of 2-(Trifluoromethyl)oxazoles from beta-Monosubstituted Enamines via Phl(OCOCF3)(2)-Mediated Trifluoroacetoxylation and Cyclization Zhao, Feifei; Liu, Xin; Qi, Rui; et al. Journal of Organic Chemistry 76
2011 Synthesis of 1,2-Diketones from beta-Keto Nitriles via a Protection-Oxidative-Decyanation-Deprotection Protocol Liu, Yu; Yun, Xiliu; Zhang-Negrerie, Daisy; et al. Synthesis-Stuttgart
2012 Synthesis of N-substituted carbazolones from alpha-iodo enaminones via Pd(0)-catalyzed intramolecular coupling under microwave irradiation Yun, Xi-Liu; Bi, Wen-Ying; Huang, Jian-Hui; et al. Tetrahedron Letters 53
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